5AMINO-10X

XENE BIOLABS RESEARCH SERIES
FOR RESEARCH USE ONLY

Category: Lipolytic Peptide | Half-life: 20-30 min

Mechanism

NNMT (Nicotinamide N-Methyltransferase) inhibitor. By inhibiting NNMT in adipose tissue, 5-Amino-1MQ increases intracellular NAD+ levels, activates SIRT1 and AMPK pathways, enhances energy expenditure, promotes fat cell shrinkage, and supports metabolic rate upregulation. No direct GH or IGF-1 effects.

Dosing Protocol

50–100 mg/day oral.

50 mg capsules:

  • 50 mg/day = 1 capsule
  • 100 mg/day = 2 capsules

Timing: Morning, with or without food.

Cycle Length: 8–12 weeks.

Critical: Daily consistency is important for optimal results. Fasting is not required. Best used alongside a calorie-controlled diet and regular exercise program to maximize metabolic and body-composition benefits.

5-Amino-1MQ

5AMINO-10X | NNMT Inhibitor / Metabolic Activator | CAS: 42464-96-0

5-Amino-1MQ is a small molecule inhibitor of nicotinamide N-methyltransferase (NNMT), an enzyme highly expressed in
adipose tissue that reduces NAD+ availability and impairs energy expenditure. By inhibiting NNMT, 5-Amino-1MQ raises
intracellular NAD+, activates SIRT1, boosts AMPK, and drives fat cell shrinkage and metabolic rate upregulation

ParameterDetails
Dose50–100 mg per day (oral)
TimingMorning, with or without food
Cycle Length8–12 weeks
Form

Capsule / Oral

STACKING RECOMMENDATIONS

Synergistic with MOTS-c (AMPK convergence), NAD+ supplementation (substrate support), Retatrutide or HGH Frag
(fat-loss amplification), and Berberine. Excellent metabolic triple-stack: 5-Amino-1MQ + MOTS-c + Berberine.

NOTE: Oral administration — most convenient in lineup. Raises NAD+ indirectly. Stack with NMN or NR for substrate augmentation